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METHYLPHENIDATE HYDROCHLORIDE

Prescription ANDA Schedule CII TE AB Official labelling
Informational index, not medical advice. Content is reproduced from public FDA and NLM data. Always confirm against the manufacturer's current prescribing information. Report adverse events to FDA MedWatch.

Overview

Brand name
METHYLPHENIDATE HYDROCHLORIDE
Generic name
Methylphenidate Hydrochloride
Dosage form
Tablet
Route
Oral
Marketing category
ANDA · ANDA
Labeler
Bryant Ranch Prepack
Product type
Human Prescription Drug
DEA schedule
CII
Active ingredients
3
NDC product codes
48
Packages
77
Data completeness
83% of corroborating sources present

Active ingredients

Source: NDC Directory
Active ingredients and strengths as listed in the NDC Directory.
Ingredient Strength RxCUI Monograph
Methylphenidate Hydrochloride 10 mg/1 1091341 View
Methylphenidate Hydrochloride 20 mg/1 1091341 View
Methylphenidate Hydrochloride 5 mg/1 1091341 View

Forms, strengths and routes

Source: NDC Directory
Dosage form
Tablet
Route of administration
Oral
Presentations
125

Pharmacologic classes are listed in the class section below.

Pharmacologic class

Source: NDC Directory
Established pharmacologic classes (EPC), mechanisms of action (MoA), chemical structures (CS) and physiologic effects (PE).
Class Type Browse
Central Nervous System Stimulant [EPC] EPC All 93 members
Central Nervous System Stimulation [PE] PE All 95 members

Regulatory status

Source: Drugs@FDANDC Directory
Application number
208737
Application type
ANDA · Abbreviated New Drug Application
Approval date
February 1, 2019
Sponsor
CEDIPROF INC
Products on application
3
Submissions recorded
3
Products approved under application 208737.
Product Trade name Form Strength Ingredient Status TE Flags
208737-001 METHYLPHENIDATE HYDROCHLORIDE TABLET METHYLPHENIDATE HYDROCHLORIDE Prescription AB
208737-002 METHYLPHENIDATE HYDROCHLORIDE TABLET METHYLPHENIDATE HYDROCHLORIDE Prescription AB
208737-003 METHYLPHENIDATE HYDROCHLORIDE TABLET METHYLPHENIDATE HYDROCHLORIDE Prescription AB

Therapeutic equivalence

Source: Orange Book
TE code
AB
Reference Listed Drug
No
Reference Standard
No

What this rating means: Therapeutically equivalent — bioequivalence demonstrated by in vivo or in vitro testing

Codes beginning with “A” indicate products the FDA considers therapeutically equivalent. Codes beginning with “B” indicate bioequivalence has not been established. See methodology.

Approval history

Source: Drugs@FDA
Most recent submissions on application 208737.
Type No. Action Status Date Review
Supplement 2 Labeling Approved April 1, 2024 Standard
Supplement 1 Labeling Approved December 16, 2022 Standard
Original application 1 Approved February 1, 2019 Standard

Prescribing information

Source: openFDA Drug Labeling

Reproduced verbatim from the Structured Product Labeling submitted to the FDA (effective 20260102). This is the manufacturer's labelling text, not a summary and not advice.

HUMAN PRESCRIPTION DRUG · 20260102 HUMAN PRESCRIPTION DRUG · 20251022 HUMAN PRESCRIPTION DRUG · 20250918 HUMAN PRESCRIPTION DRUG · 20250317

Boxed Warning

openFDA Drug Labeling

WARNING: ABUSE, MISUSE, AND ADDICTION WARNING: ABUSE, MISUSE, AND ADDICTION Methylphenidate hydrochloride tablets have a high potential for abuse and misuse, which can lead to the development of a substance use disorder, including addiction. Misuse and abuse of CNS stimulants, including methylphenidate hydrochloride tablets, can result in overdose and death [see Overdosage (10) ] , and this risk is increased with higher doses or unapproved methods of administration, such as snorting or injection. Before prescribing methylphenidate hydrochloride tablets, assess each patient’s risk for abuse, misuse, and addiction. Educate patients and their families about these risks, proper storage of the drug, and proper disposal of any unused drug. Throughout methylphenidate hydrochloride tablets treatment, reassess each patient’s risk of abuse, misuse, and addiction and frequently monitor for signs and symptoms of abuse, misuse, and addiction [see Warnings and Precautions (5.1) and Drug Abuse and Dependence (9.2) ] . WARNING: ABUSE, MISUSE, AND ADDICTION See full prescribing information for complete boxed warning. Methylphenidate hydrochloride tablets have a high potential for abuse and misuse, which can lead to the development of a substance use disorder, including addiction. Misuse and abuse of CNS stimulants, including methylphenidate hydrochloride tablets, can result in overdose and death (5.1 , 9.2 , 10) : Before prescribing methylphenidate hydrochloride tablets, assess each patient’s risk for abuse, misuse, and addiction. Educate patients and their families about these risks, proper storage of the drug, and proper disposal of any unused drug. Throughout treatment, reassess each patient’s risk and frequently monitor for signs and symptoms of abuse, misuse, and addiction.

Recent Major Changes

openFDA Drug Labeling

Boxed Warning 10/2023 Dosage and Administration (2.1) 10/2023 Warnings and Precautions (5.1, 5.2, 5.8, 5.9, 5.10) 10/2023 Boxed Warning 10/2023 Dosage and Administration ( 2.1 ) 10/2023 Warnings and Precautions ( 5.1 , 5.2 , 5.8 , 5.9 , 5.10 ) 10/2023

Indications and Usage

openFDA Drug Labeling

1 INDICATIONS AND USAGE Methylphenidate hydrochloride tablets are indicated for the treatment of: • Attention Deficit Hyperactivity Disorders (ADHD) in pediatric patients 6 years and older and adults • Narcolepsy Methylphenidate hydrochloride tablets are a central nervous system (CNS) stimulant indicated for the treatment of Attention Deficit Hyperactivity Disorders (ADHD) and Narcolepsy ( 1 ).

Dosage and Administration

openFDA Drug Labeling

2. DOSAGE AND ADMINISTRATION Methylphenidate Hydrochloride Tablets, USP (2.2) : Pediatric Patients 6 Years and Older: Start with 5 mg twice daily (before breakfast and lunch), titrating the dose weekly in 5- to 10- mg increments. Dosages above 60 mg/day are not recommended. Adults: Average daily dosage is 20 mg to 30 mg, administered 2 or 3 times daily, preferably 30 to 45 minutes before meals. Maximum total daily dosage is 60 mg. 2.1 Pretreatment Screening Prior to treating pediatric patients and adults with central nervous system (CNS) stimulants, including methylphenidate hydrochloride tablets, assess for the presence of cardiac disease (i.e., perform a careful history, including family history of sudden death or ventricular arrhythmia, and physical examination) [see Warnings and Precautions (5.2)] . Assess the risk of abuse prior to prescribing, and monitor for signs of abuse and dependence while on therapy. Maintain careful prescription records, educate patients about abuse, monitor for signs of abuse and overdose, and periodically reevaluate the need for methylphenidate hydrochloride tablets use [see Boxed Warning, Warnings and Precautions (5.1), Drug Abuse and Dependence (9.2, 9.3)]. 2.2 General Dosing Information Methylphenidate Hydrochloride Tablets Pediatric Patients 6 years and Older: Start with 5 mg orally twice daily (before breakfast and lunch). Increase dosage gradually, in increments of 5- to 10- mg weekly. Daily dosage above 60 mg is not recommended. Adults: Average dosage is 20 to 30 mg daily. Administer orally in divided doses 2 or 3 times daily, preferably 30 to 45 minutes before meals. Maximum total daily dosage is 60 mg. Patients who are unable to sleep if medication is taken late in the day should take the last dose before 6 p.m. Pharmacological treatment of ADHD may be needed for extended periods. Periodically reevaluate the long-term use of methylphenidate hydrochloride tablets, and adjust dosage as needed. 2.3 Dose Reduction and Discontinuation If paradoxical worsening of symptoms or other adverse reactions occur, reduce the dosage, or, if necessary, discontinue methylphenidate hydrochloride tablets. If improvement is not observed after appropriate dosage adjustment over a one-month period, the drug should be discontinued.

Dosage Forms and Strengths

openFDA Drug Labeling

3 DOSAGE FORMS AND STRENGTHS Methylphenidate Hydrochloride Tablets, USP 5 mg, light purple, round-shaped, flat faced, beveled edge, uncoated tablets, debossed with "228" on one side and S5 on the other side. 10 mg, light green, round-shaped, flat faced, beveled edge, uncoated tablets, debossed with "229" on one side and S and 10 on either side of the score line on the other side. 20 mg, light peach, round-shaped, flat faced, beveled edge, uncoated tablets, debossed with "230" on one side and S and 20 on either side of the score line on the other side. Tablets: 5 mg, 10 mg, and 20 mg (3)

Contraindications

openFDA Drug Labeling

2.3 Dosage Reduction and Discontinuation If paradoxical worsening of symptoms or other adverse reactions occur, reduce the dosage, or, if necessary, discontinue methylphenidate hydrochloride tablets. If improvement is not observed after appropriate dosage adjustment over a one-month period, the drug should be discontinued.

4 CONTRAINDICATIONS • Hypersensitivity to methylphenidate or other components of methylphenidate hydrochloride tablets. Hypersensitivity reactions, such as angioedema and anaphylactic reactions, have been reported in patients treated with methylphenidate [see Adverse Reactions ( 6 )] . • Concomitant treatment with monoamine oxidase inhibitors (MAOIs), or within 14 days following discontinuation of treatment with an MAOI, because of the risk of hypertensive crises [see Drug Interactions ( 7.1 )] . • Known hypersensitivity to methylphenidate or other product components of methylphenidate hydrochloride tablets ( 4 ). • Concurrent treatment with a monoamine oxidase inhibitor (MAOI), or use of an MAOI within the preceding 14 days ( 4 ).

Warnings and Cautions

openFDA Drug Labeling

5 WARNINGS AND PRECAUTIONS Risks to Patients with Serious Cardiac Disease : Avoid use in patients with known structural cardiac abnormalities, cardiomyopathy, serious cardiac arrhythmias, coronary artery disease, or other serious cardiac disease (5.2). Increased Blood Pressure and Heart Rate : Monitor blood pressure and pulse (5.3). Psychiatric Adverse Reactions : Prior to initiating methylphenidate hydrochloride tablets, screen patients for risk factors for developing a manic episode. If new psychotic or manic symptoms occur, consider discontinuing methylphenidate hydrochloride tablets (5.4). Priapism : If abnormally sustained or frequent and painful erections occur, patients should seek immediate medical attention (5.5). Peripheral Vasculopathy, Including Raynaud’s Phenomenon : Careful observation for digital changes is necessary during methylphenidate hydrochloride tablets treatment. Further clinical evaluation (e.g., rheumatology referral) may be appropriate for patients who develop signs or symptoms of peripheral vasculopathy (5.6). Long-Term Suppression of Growth in Pediatric Patients : Closely monitor growth (height and weight) in pediatric patients. Pediatric patients not growing or gaining height or weight as expected may need to have their treatment interrupted (5.7). Acute Angle Closure Glaucoma: Methylphenidate hydrochloride tablets -treated patients considered at risk for acute angle closure glaucoma (e.g., patients with significant hyperopia) should be evaluated by an ophthalmologist (5.8). Increased Intraocular Pressure (IOP) and Glaucoma: Prescribe methylphenidate hydrochloride tablets to patients with open-angle glaucoma or abnormally increased IOP only if the benefit of treatment is considered to outweigh the risk. Closely monitor patients with a history of increased IOP or open angle glaucoma (5.9). Motor and Verbal Tics, and Worsening of Tourette’s Syndrome: Before initiating methylphenidate hydrochloride tablets, assess the family history and clinically evaluate patients for tics or Tourette’s syndrome. Regularly monitor patients for the emergence or worsening of tics or Tourette’s syndrome. Discontinue treatment if clinically appropriate (5.10). 5.1 Abuse, Misuse, and Addiction Methylphenidate hydrochloride tablets have a high potential for abuse and misuse. The use of methylphenidate hydrochloride tablets exposes individuals to the risks of abuse and misuse, which can lead to the development of a substance use disorder, including addiction. Methylphenidate hydrochloride tablets can be diverted for nonmedical use into illicit channels or distribution [see Drug Abuse and Dependence (9.2) ]. Misuse and abuse of CNS stimulants, including methylphenidate hydrochloride tablets, can result in overdose and death [see Overdosage (10)] , and this risk is increased with higher doses or unapproved methods of administration, such as snorting or injection. Before prescribing methylphenidate hydrochloride tablets, assess each patient’s risk for abuse, misuse, and addiction. Educate patients and their families about these risks and proper disposal of any unused drug. Advise patients to store methylphenidate hydrochloride tablets in a safe place, preferably locked, and instruct patients to not give methylphenidate hydrochloride tablets to anyone else. Throughout methylphenidate hydrochloride tablets treatment, reassess each patient’s risk of abuse, misuse, and addiction and frequently monitor for signs and symptoms of abuse, misuse, and addiction. 5.2 Risks to Patients with Serious Cardiac Disease Sudden death has been reported in patients with structural cardiac abnormalities or other serious cardiac disease who are treated with CNS stimulants at the recommended ADHD dosage. Avoid methylphenidate hydrochloride tablets use in patients with known serious structural cardiac abnormalities, cardiomyopathy, serious cardiac arrhythmia, coronary artery disease, or other serious cardiac disease. 5.3 Increased Blood Pressure and …

Adverse Reactions

openFDA Drug Labeling

6 ADVERSE REACTIONS The following are discussed in more detail in other sections of the labeling: • Abuse, Misuse, and Addiction [see Boxed Warning , Warnings and Precautions ( 5.1 ), Drug Abuse and Dependence ( 9.2 , 9.3 ) ] • Known hypersensitivity to methylphenidate or other ingredients of methylphenidate hydrochloride tablets [see Contraindications ( 4 )] • Hypertensive crisis with Concomitant Use of Monoamine Oxidase Inhibitors [see Contraindications ( 4 ), Drug Interactions ( 7.1 )] • Risks to Patients with Serious Cardiac Disease [see Warnings and Precautions ( 5.2 )] • Increased Blood Pressure and Heart Rate [see Warnings and Precautions ( 5.3 )] • Psychiatric Adverse Reactions [see Warnings and Precautions ( 5.4 )] • Priapism [see Warnings and Precautions ( 5.5 )] • Peripheral Vasculopathy, Including Raynaud’s Phenomenon [see Warnings and Precautions ( 5.6 )] • Long-Term Suppression of Growth in Pediatric Patients [see Warnings and Precautions ( 5.7 )] • Acute Angle Closure Glaucoma [see Warnings and Precautions ( 5.8 )] • Increased Intraocular Pressure and Glaucoma [see Warnings and Precautions ( 5.9 )] • Motor and Verbal Tics, and Worsening of Tourette’s Syndrome [see Warnings and Precautions ( 5.10 )] The following adverse reactions associated with the use of methylphenidate hydrochloride tablets and other methylphenidate products were identified in clinical trials, spontaneous reports, and literature. Because these reactions were reported voluntarily from a population of uncertain size, it is not always possible to estimate their frequency reliably or to establish a causal relationship to drug exposure. Adverse Reactions Reported with Methylphenidate Hydrochloride Tablets Infections and Infestations: nasopharyngitis Blood and the Lymphatic System Disorders : leukopenia, thrombocytopenia, anemia Immune System Disorders: hypersensitivity reactions, including angioedema, and anaphylaxis Metabolism and Nutrition Disorders: decreased appetite, reduced weight gain, and suppression of growth during prolonged use in pediatric patients Psychiatric Disorders: insomnia, anxiety, restlessness, agitation, psychosis (sometimes with visual and tactile hallucinations), depressed mood, depression Nervous System Disorders: headache, dizziness, tremor, dyskinesia, including choreoathetoid movements, drowsiness, convulsions, cerebrovascular disorders (including vasculitis, cerebral hemorrhages and cerebrovascular accidents), serotonin syndrome in combination with serotonergic drugs Eye Disorders: blurred vision, difficulties in visual accommodation Cardiac Disorders: tachycardia, palpitations, increased blood pressure, arrhythmias, angina pectoris Respiratory, Thoracic, and Mediastinal Disorders: cough Gastrointestinal Disorders: dry mouth, nausea, vomiting, abdominal pain, dyspepsia Hepatobiliary Disorders: abnormal liver function, ranging from transaminase elevation to severe hepatic injury Skin and Subcutaneous Tissue Disorders: hyperhidrosis, pruritus, urticaria, exfoliative dermatitis, scalp hair loss, erythema multiforme rash, thrombocytopenic purpura Musculoskeletal and Connective Tissue Disorders: arthralgia, muscle cramps, rhabdomyolysis, trismus Investigations: weight loss (adult ADHD patients) Vascular Disorders: peripheral coldness, Raynaud's phenomenon Additional Adverse Reactions Reported with Other Methylphenidate-Containing Products The list below shows adverse reactions not listed for methylphenidate hydrochloride tablets that have been reported with other methylphenidate-containing products. Blood and Lymphatic Disorders: pancytopenia Immune System Disorders: hypersensitivity reactions, such as auricular swelling, bullous conditions, eruptions, exanthemas Psychiatric Disorders: affect lability, mania, disorientation, and libido changes Nervous System Disorders: migraine, motor and verbal tics Eye Disorders: diplopia, increased intraocular pressure, mydriasis Cardiac Disorders: sudden cardiac death, myocardial infarc …

Drug Interactions

openFDA Drug Labeling

7 DRUG INTERACTIONS Antihypertensive Drugs: Monitor blood pressure. Adjust dosage of antihypertensive drug as needed (7.1). Halogenated Anesthetics: Avoid use of methylphenidate hydrochloride tablets on the day of surgery if halogenated anesthetics will be used (7.1). 7.1 Clinically Important Drug Interactions with Methylphenidate Hydrochloride Table 1 presents clinically important drug interactions with methylphenidate hydrochloride tablets Table 1: Clinically Important Drug Interactions with Methylphenidate Hydrochloride Monoamine Oxidase Inhibitors (MAOI) Clinical Impact Concomitant use of MAOIs and CNS stimulants, including methylphenidate hydrochloride can cause hypertensive crisis. Potential outcomes include death, stroke, myocardial infarction, aortic dissection, ophthalmological complications, eclampsia, pulmonary edema, and renal failure [see Contraindications (4)]. Intervention Concomitant use of methylphenidate hydrochloride with MAOIs or within 14 days after discontinuing MAOI treatment is contraindicated. Examples selegiline, tranylcypromine, isocarboxazid, phenelzine, linezolid, methylene blue Antihypertensive Drugs Clinical Impact Methylphenidate hydrochloride may decrease the effectiveness of drugs used to treat hypertension [see Warnings and Precautions (5.3)] . Intervention Monitor blood pressure and adjust the dosage of the antihypertensive drug as needed. Examples Potassium-sparing and thiazide diuretics, calcium channel blockers, angiotensin-converting-enzyme (ACE) inhibitors, angiotensin II receptor blockers (ARBs), beta blockers, centrally acting alpha-2 receptor agonists Halogenated Anesthetics Clinical Impact Concomitant use of halogenated anesthetics and methylphenidate hydrochloride may increase the risk of sudden blood pressure and heart rate increase during surgery. Intervention Avoid use of methylphenidate hydrochloride in patients being treated with anesthetics on the day of surgery. Examples halothane, isoflurane, enflurane, desflurane, sevoflurane Risperidone Clinical Impact Combined use of methylphenidate with risperidone when there is a change, whether an increase or decrease, in dosage of either or both medications, may increase the risk of extrapyramidal symptoms (EPS) Intervention Monitor for signs of EPS

Use in Specific Populations

openFDA Drug Labeling

8 USE IN SPECIFIC POPULATIONS 8.1 Pregnancy Pregnancy Exposure Registry There is a pregnancy exposure registry that monitors pregnancy outcomes in women exposed to ADHD medications, including Methylphenidate hydrochloride tablets, during pregnancy. Healthcare providers are encouraged to register patients by calling the National Pregnancy Registry for ADHD Medications at 1-866-961-2388 or visiting https://womensmentalhealth.org/adhd-medications/. Risk Summary Published studies and postmarketing reports on methylphenidate use during pregnancy have not identified a drug-associated risk of major birth defects, miscarriage or adverse maternal or fetal outcomes. There may be risks to the fetus associated with the use of CNS stimulants use during pregnancy (see Clinical Considerations) . No effects on morphological development were observed in embryo-fetal development studies with oral administration of methylphenidate to pregnant rats and rabbits during organogenesis at doses up to 10 and 15 times, respectively, the maximum recommended human dose (MRHD) of 60 mg/day given to adolescents on a mg/m 2 basis. However, spina bifida was observed in rabbits at a dose 52 times the MRHD given to adolescents. A decrease in pup body weight was observed in a pre- and post-natal development study with oral administration of methylphenidate to rats throughout pregnancy and lactation at doses 6 times the MRHD given to adolescents (see Data) . The estimated background risk of major birth defects and miscarriage for the indicated population is unknown. All pregnancies have a background risk of birth defect, loss, or other adverse outcomes. In the U.S. general population, the estimated background risk of major birth defects and miscarriage in clinically recognized pregnancies is 2% to 4% and 15% to 20%, respectively. Clinical Considerations Fetal/Neonatal Adverse Reactions CNS stimulants, such as Methylphenidate hydrochloride tablets, can cause vasoconstriction and thereby decrease placental perfusion. No fetal and/or neonatal adverse reactions have been reported with the use of therapeutic doses of methylphenidate during pregnancy; however, premature delivery and low birth weight infants have been reported in amphetamine-dependent mothers. Data Animal Data In embryo-fetal development studies conducted in rats and rabbits, methylphenidate was administered orally at doses of up to 75 and 200 mg/kg/day, respectively, during the period of organogenesis. Malformations (increased incidence of fetal spina bifida) were observed in rabbits at the highest dose, which is approximately 52 times the MRHD of 60 mg/day given to adolescents on a mg/m 2 basis. The no effect level for embryo-fetal development in rabbits was 60 mg/kg/day (15times the MRHD given to adolescents on a mg/m 2 basis). There was no evidence of morphological development effects in rats, although increased incidences of fetal skeletal variations were seen at the highest dose level (10 times the MRHD of 60 mg/day given to adolescents on a mg/m 2 basis), which was also maternally toxic. The no effect level for embryo-fetal development in rats was 25 mg/kg/day (3 times the MRHD on a mg/m 2 basis). When methylphenidate was administered to rats throughout pregnancy and lactation at doses of up to 45 mg/kg/day, offspring body weight gain was decreased at the highest dose (6 times the MRHD of 60 mg/day given to adolescents on a mg/m2 basis), but no other effects on postnatal development were observed. The no effect level for pre- and postnatal development in rats was 15 mg/kg/day (approximately 2 times the MRHD given to adolescents on a mg/m 2 basis). 8.2 Lactation Risk Summary Limited published literature, based on milk sampling from seven mothers reports that methylphenidate is present in human milk, which resulted in infant doses of 0.16% to 0.7% of the maternal weight-adjusted dosage and a milk/plasma ratio ranging between 1.1 and 2.7. There are no reports of adverse effects on the breastfed infa …

Mechanism of Action

openFDA Drug Labeling

12.1 Mechanism of Action Methylphenidate hydrochloride is a central nervous system (CNS) stimulant. The mode of therapeutic action in ADHD and narcolepsy is not known.

Description

openFDA Drug Labeling

11 DESCRIPTION Methylphenidate hydrochloride tablets contain methylphenidate hydrochloride, USP a CNS stimulant. It is available as tablets of 5 mg, 10 mg, and 20 mg strengths for oral administration. Methylphenidate hydrochloride is methyl α-phenyl-2-piperidineacetate hydrochloride, and its structural formula is: Methylphenidate hydrochloride, USP is a white, odorless, fine crystalline powder. Its solutions are acid to litmus. It is freely soluble in water and in methanol, soluble in alcohol, and slightly soluble in chloroform and in acetone. Its molecular weight is 269.77 g/mol. Each tablet contains 5 mg, 10 mg, or 20 mg of methylphenidate hydrochloride, USP. Inactive ingredients include: lactose monohydrate, magnesium stearate, polyethylene glycol 8000, and talc. In addition, the 5 mg tablet contains FD&C blue No. 2 aluminum lake and FD&C red No. 40 aluminum lake, the 10 mg tablet contains FD&C blue No. 2 aluminum lake and D&C yellow No. 10 aluminum lake and the 20 mg tablet contains FD&C yellow No. 6 aluminum lake. Structure

10 OVERDOSAGE Clinical Effects of Overdose Overdose of CNS stimulants is characterized by the following sympathomimetic effects: • Cardiovascular effects including tachyarrhythmias, and hypertension or hypotension. Vasospasm, myocardial infarction, or aortic dissection may precipitate sudden cardiac death. Takotsubo cardiomyopathy may develop. • CNS effects including psychomotor agitation, confusion, and hallucinations. Serotonin syndrome, seizures, cerebral vascular accidents, and coma may occur. • Life-threatening hyperthermia (temperatures greater than 104°F) and rhabdomyolysis may develop. Overdose Management Consider the possibility of multiple drug ingestion. Because methylphenidate has a large volume of distribution and is rapidly metabolized, dialysis is not useful. Consider contacting the Poison Help line (1-800-222-1222) or a medical toxicologist for additional overdose management recommendations.

How Supplied / Storage and Handling

openFDA Drug Labeling

16 HOW SUPPLIED/STORAGE AND HANDLING Methylphenidate Hydrochloride Tablets, USP are available as follows 5 mg Tablets - light yellow colored, round, flat face tablets with "n above 573" debossed on one side and plain on the other side, supplied as: Bottles of 30 .........................................NDC 43386-573-03 Bottles of 100.......................................NDC 43386-573-01 Bottles of 500 .......................................NDC 43386-573-05 10 mg Tablets - white to off white colored, round, flat face tablets with "n above 574" debossed on one side and bisected line debossed on the other side, supplied as: Bottles of 30 ....................................... NDC 43386-574-03 Bottles of 100.......................................NDC 43386-574-01 Bottles of 500 .......................................NDC 43386-574-05 20 mg Tablets - light yellow colored, round biconvex tablets with "n above 575" debossed on one side and bisect line debossed on the other side, supplied as: Bottles of 30 .........................................NDC 43386-575-03 Bottles of 100.......................................NDC 43386-575-01 Bottles of 500 .......................................NDC 43386-575-05 Store at 20°C to 25°C (68°F to 77°F), excursions permitted between 15oC and 30oC (59oF and 86oF) [see USP Controlled Room Temperature]. Protect from light. Dispense in tight, light-resistant container (USP). Disposal Comply with local laws and regulations on drug disposal of CNS stimulants. Dispose of remaining, unused, or expired methylphenidate hydrochloride tablets by a medicine takeback program or by an authorized collector registered with the Drug Enforcement Administration. If no take-back program or authorized collector is available, mix methylphenidate hydrochloride tablets with an undesirable, nontoxic substance to make it less appealing to children and pets. Place the mixture in a container, such as a sealed plastic bag and discard methylphenidate hydrochloride tablets in the household trash.

Adverse event reports

Source: openFDA FAERS
58,466
FAERS reports mentioning this drug
as of 2026-09-25T03:42:24+00:00
A report count is not a risk measure. FAERS accepts voluntary and mandatory reports without establishing causation, and reporting is influenced by how widely a drug is used, how long it has been marketed, and media attention. FDA states that reports “do not prove that the drug caused the event”. Compare rates, not totals.

Attributed to this product's most-reported active ingredient: METHYLPHENIDATE HYDROCHLORIDE. Combination products with more than six active ingredients are not attributed, because a report count summed across a long ingredient list measures the list, not the medicine.

Recalls

Source: FDA Enforcement
Drug recall enforcement reports associated with this product.
Classification Reported Firm Reason Status
Class II August 2, 2023 SUN PHARMACEUTICAL INDUSTRIES INC Presence of Foreign Substance: Metal embedded in a tablet. Terminated

Packaging and NDCs

Source: NDC Directory
Every National Drug Code package associated with this medication. The NDC is the identifier used for dispensing, billing and pharmacovigilance in the United States.
Package NDC Product NDC Labeler Description Marketing start
16729-478-01 16729-478 Accord Healthcare, Inc. 100 TABLET in 1 BOTTLE (16729-478-01) December 23, 2020
16729-479-01 16729-479 Accord Healthcare, Inc. 100 TABLET in 1 BOTTLE (16729-479-01) December 17, 2020
16729-480-01 16729-480 Accord Healthcare, Inc. 100 TABLET in 1 BOTTLE (16729-480-01) December 17, 2020
68084-805-21 68084-805 American Health Packaging 30 BLISTER PACK in 1 BOX, UNIT-DOSE (68084-805-21) / 1 TABLET in 1 BLISTER PACK (68084-805-11) September 30, 2014
68084-823-21 68084-823 American Health Packaging 30 BLISTER PACK in 1 BOX, UNIT-DOSE (68084-823-21) / 1 TABLET in 1 BLISTER PACK (68084-823-11) September 30, 2014
0115-1800-01 0115-1800 Amneal Pharmaceuticals of New York LLC 100 TABLET in 1 BOTTLE, PLASTIC (0115-1800-01) April 7, 2014
0115-1801-01 0115-1801 Amneal Pharmaceuticals of New York LLC 100 TABLET in 1 BOTTLE, PLASTIC (0115-1801-01) April 7, 2014
0115-1802-01 0115-1802 Amneal Pharmaceuticals of New York LLC 100 TABLET in 1 BOTTLE, PLASTIC (0115-1802-01) April 7, 2014
67877-616-01 67877-616 Ascend Laboratories, LLC 100 TABLET in 1 BOTTLE (67877-616-01) October 6, 2019
67877-616-33 67877-616 Ascend Laboratories, LLC 10 BLISTER PACK in 1 CARTON (67877-616-33) / 1 TABLET in 1 BLISTER PACK October 6, 2019
67877-617-01 67877-617 Ascend Laboratories, LLC 100 TABLET in 1 BOTTLE (67877-617-01) October 6, 2019
67877-617-33 67877-617 Ascend Laboratories, LLC 10 BLISTER PACK in 1 CARTON (67877-617-33) / 1 TABLET in 1 BLISTER PACK October 6, 2019
67877-618-01 67877-618 Ascend Laboratories, LLC 100 TABLET in 1 BOTTLE (67877-618-01) October 6, 2019
67877-618-33 67877-618 Ascend Laboratories, LLC 10 BLISTER PACK in 1 CARTON (67877-618-33) / 1 TABLET in 1 BLISTER PACK October 6, 2019
13107-380-01 13107-380 Aurolife Pharma, LLC 100 TABLET in 1 BOTTLE (13107-380-01) April 11, 2017
13107-381-01 13107-381 Aurolife Pharma, LLC 100 TABLET in 1 BOTTLE (13107-381-01) April 11, 2017
13107-382-01 13107-382 Aurolife Pharma, LLC 100 TABLET in 1 BOTTLE (13107-382-01) April 11, 2017
63629-1172-1 63629-1172 Bryant Ranch Prepack 100 TABLET in 1 BOTTLE (63629-1172-1) August 16, 2013
71335-1219-1 71335-1219 Bryant Ranch Prepack 30 TABLET in 1 BOTTLE (71335-1219-1) October 31, 2024
71335-1219-2 71335-1219 Bryant Ranch Prepack 100 TABLET in 1 BOTTLE (71335-1219-2) October 31, 2024
71335-1219-3 71335-1219 Bryant Ranch Prepack 90 TABLET in 1 BOTTLE (71335-1219-3) April 24, 2019
71335-1219-4 71335-1219 Bryant Ranch Prepack 60 TABLET in 1 BOTTLE (71335-1219-4) April 24, 2019
71335-1219-5 71335-1219 Bryant Ranch Prepack 120 TABLET in 1 BOTTLE (71335-1219-5) October 31, 2024
71335-2968-1 71335-2968 Bryant Ranch Prepack 100 TABLET in 1 BOTTLE (71335-2968-1) November 11, 2025
72162-1636-1 72162-1636 Bryant Ranch Prepack 100 TABLET in 1 BOTTLE (72162-1636-1) August 16, 2013
72162-2019-1 72162-2019 Bryant Ranch Prepack 100 TABLET in 1 BOTTLE (72162-2019-1) April 3, 2024
72162-2019-6 72162-2019 Bryant Ranch Prepack 60 TABLET in 1 BOTTLE (72162-2019-6) April 3, 2024
72162-2086-1 72162-2086 Bryant Ranch Prepack 100 TABLET in 1 BOTTLE (72162-2086-1) April 3, 2024
72162-2087-1 72162-2087 Bryant Ranch Prepack 100 TABLET in 1 BOTTLE (72162-2087-1) April 3, 2024
72162-2428-1 72162-2428 Bryant Ranch Prepack 100 TABLET in 1 BOTTLE (72162-2428-1) November 18, 2024
72162-2429-1 72162-2429 Bryant Ranch Prepack 100 TABLET in 1 BOTTLE (72162-2429-1) November 18, 2024
72162-2430-1 72162-2430 Bryant Ranch Prepack 100 TABLET in 1 BOTTLE (72162-2430-1) November 18, 2024
31722-173-01 31722-173 Camber Pharmaceutical Inc 100 TABLET in 1 BOTTLE (31722-173-01) October 1, 2015
31722-173-05 31722-173 Camber Pharmaceutical Inc 500 TABLET in 1 BOTTLE (31722-173-05) October 1, 2015
31722-174-01 31722-174 Camber Pharmaceutical Inc 100 TABLET in 1 BOTTLE (31722-174-01) October 1, 2015
31722-174-05 31722-174 Camber Pharmaceutical Inc 500 TABLET in 1 BOTTLE (31722-174-05) October 1, 2015
31722-175-01 31722-175 Camber Pharmaceutical Inc 100 TABLET in 1 BOTTLE (31722-175-01) October 1, 2015
31722-175-05 31722-175 Camber Pharmaceutical Inc 500 TABLET in 1 BOTTLE (31722-175-05) October 1, 2015
10702-100-01 10702-100 KVK-TECH, INC. 100 TABLET in 1 BOTTLE (10702-100-01) May 11, 2017
10702-101-01 10702-101 KVK-TECH, INC. 100 TABLET in 1 BOTTLE (10702-101-01) May 11, 2017
10702-102-01 10702-102 KVK-TECH, INC. 100 TABLET in 1 BOTTLE (10702-102-01) May 11, 2017
43386-573-01 43386-573 Lupin Pharmaceuticals,Inc. 100 TABLET in 1 BOTTLE (43386-573-01) January 20, 2016
43386-574-01 43386-574 Lupin Pharmaceuticals,Inc. 100 TABLET in 1 BOTTLE (43386-574-01) January 20, 2016
43386-575-01 43386-575 Lupin Pharmaceuticals,Inc. 100 TABLET in 1 BOTTLE (43386-575-01) January 20, 2016
75834-324-01 75834-324 Nivagen Pharmaceuticals, Inc. 100 TABLET in 1 BOTTLE (75834-324-01) April 16, 2024
75834-325-01 75834-325 Nivagen Pharmaceuticals, Inc. 100 TABLET in 1 BOTTLE (75834-325-01) April 16, 2024
75834-326-01 75834-326 Nivagen Pharmaceuticals, Inc. 100 TABLET in 1 BOTTLE (75834-326-01) April 16, 2024
43547-486-10 43547-486 Solco Healthcare US,LLC 100 TABLET in 1 BOTTLE (43547-486-10) July 1, 2020
43547-487-10 43547-487 Solco Healthcare US,LLC 100 TABLET in 1 BOTTLE (43547-487-10) July 1, 2020
43547-488-10 43547-488 Solco Healthcare US,LLC 100 TABLET in 1 BOTTLE (43547-488-10) July 1, 2020
0406-1142-01 0406-1142 SpecGx LLC 100 TABLET in 1 BOTTLE (0406-1142-01) November 27, 1998
0406-1142-10 0406-1142 SpecGx LLC 1000 TABLET in 1 BOTTLE (0406-1142-10) November 27, 1998
0406-1144-01 0406-1144 SpecGx LLC 100 TABLET in 1 BOTTLE (0406-1144-01) November 27, 1998
0406-1144-10 0406-1144 SpecGx LLC 1000 TABLET in 1 BOTTLE (0406-1144-10) November 27, 1998
0406-1146-01 0406-1146 SpecGx LLC 100 TABLET in 1 BOTTLE (0406-1146-01) November 27, 1998
0406-1146-10 0406-1146 SpecGx LLC 1000 TABLET in 1 BOTTLE (0406-1146-10) November 27, 1998
57664-228-08 57664-228 Sun Pharmaceutical Industries, Inc. 100 TABLET in 1 BOTTLE (57664-228-08) August 16, 2013
57664-228-13 57664-228 Sun Pharmaceutical Industries, Inc. 500 TABLET in 1 BOTTLE (57664-228-13) August 16, 2013
57664-228-18 57664-228 Sun Pharmaceutical Industries, Inc. 1000 TABLET in 1 BOTTLE (57664-228-18) August 16, 2013
57664-228-83 57664-228 Sun Pharmaceutical Industries, Inc. 30 TABLET in 1 BOTTLE (57664-228-83) August 16, 2013
57664-228-88 57664-228 Sun Pharmaceutical Industries, Inc. 100 TABLET in 1 BOTTLE (57664-228-88) August 16, 2013
57664-229-08 57664-229 Sun Pharmaceutical Industries, Inc. 100 TABLET in 1 BOTTLE (57664-229-08) August 16, 2013
57664-229-13 57664-229 Sun Pharmaceutical Industries, Inc. 500 TABLET in 1 BOTTLE (57664-229-13) August 16, 2013
57664-229-18 57664-229 Sun Pharmaceutical Industries, Inc. 1000 TABLET in 1 BOTTLE (57664-229-18) August 16, 2013
57664-229-83 57664-229 Sun Pharmaceutical Industries, Inc. 30 TABLET in 1 BOTTLE (57664-229-83) August 16, 2013
57664-229-88 57664-229 Sun Pharmaceutical Industries, Inc. 100 TABLET in 1 BOTTLE (57664-229-88) August 16, 2013
57664-230-08 57664-230 Sun Pharmaceutical Industries, Inc. 100 TABLET in 1 BOTTLE (57664-230-08) August 16, 2013
57664-230-13 57664-230 Sun Pharmaceutical Industries, Inc. 500 TABLET in 1 BOTTLE (57664-230-13) August 16, 2013
57664-230-18 57664-230 Sun Pharmaceutical Industries, Inc. 1000 TABLET in 1 BOTTLE (57664-230-18) August 16, 2013
57664-230-83 57664-230 Sun Pharmaceutical Industries, Inc. 30 TABLET in 1 BOTTLE (57664-230-83) August 16, 2013
57664-230-88 57664-230 Sun Pharmaceutical Industries, Inc. 100 TABLET in 1 BOTTLE (57664-230-88) August 16, 2013
72865-122-01 72865-122 XLCare Pharmaceuticals Inc 100 TABLET in 1 BOTTLE (72865-122-01) February 26, 2020
72865-122-05 72865-122 XLCare Pharmaceuticals Inc 500 TABLET in 1 BOTTLE (72865-122-05) February 26, 2020
72865-123-01 72865-123 XLCare Pharmaceuticals Inc 100 TABLET in 1 BOTTLE (72865-123-01) February 26, 2020
72865-123-05 72865-123 XLCare Pharmaceuticals Inc 500 TABLET in 1 BOTTLE (72865-123-05) February 26, 2020
72865-124-01 72865-124 XLCare Pharmaceuticals Inc 100 TABLET in 1 BOTTLE (72865-124-01) February 26, 2020
72865-124-05 72865-124 XLCare Pharmaceuticals Inc 500 TABLET in 1 BOTTLE (72865-124-05) February 26, 2020
16729-478 16729-478 Accord Healthcare, Inc. — December 23, 2020
16729-479 16729-479 Accord Healthcare, Inc. — December 17, 2020
16729-480 16729-480 Accord Healthcare, Inc. — December 17, 2020
68084-805 68084-805 American Health Packaging — September 30, 2014
68084-823 68084-823 American Health Packaging — September 30, 2014
0115-1800 0115-1800 Amneal Pharmaceuticals of New York LLC — April 7, 2014
0115-1801 0115-1801 Amneal Pharmaceuticals of New York LLC — April 7, 2014
0115-1802 0115-1802 Amneal Pharmaceuticals of New York LLC — April 7, 2014
67877-616 67877-616 Ascend Laboratories, LLC — October 6, 2019
67877-617 67877-617 Ascend Laboratories, LLC — October 6, 2019
67877-618 67877-618 Ascend Laboratories, LLC — October 6, 2019
13107-380 13107-380 Aurolife Pharma, LLC — April 11, 2017
13107-381 13107-381 Aurolife Pharma, LLC — April 11, 2017
13107-382 13107-382 Aurolife Pharma, LLC — April 11, 2017
63629-1172 63629-1172 Bryant Ranch Prepack — August 16, 2013
71335-1219 71335-1219 Bryant Ranch Prepack — October 1, 2015
71335-2968 71335-2968 Bryant Ranch Prepack — April 16, 2024
72162-1636 72162-1636 Bryant Ranch Prepack — August 16, 2013
72162-2019 72162-2019 Bryant Ranch Prepack — April 7, 2014
72162-2086 72162-2086 Bryant Ranch Prepack — April 7, 2014
72162-2087 72162-2087 Bryant Ranch Prepack — April 7, 2014
72162-2428 72162-2428 Bryant Ranch Prepack — April 16, 2024
72162-2429 72162-2429 Bryant Ranch Prepack — April 16, 2024
72162-2430 72162-2430 Bryant Ranch Prepack — April 16, 2024
31722-173 31722-173 Camber Pharmaceutical Inc — October 1, 2015
31722-174 31722-174 Camber Pharmaceutical Inc — October 1, 2015
31722-175 31722-175 Camber Pharmaceutical Inc — October 1, 2015
10702-100 10702-100 KVK-TECH, INC. — May 11, 2017
10702-101 10702-101 KVK-TECH, INC. — May 11, 2017
10702-102 10702-102 KVK-TECH, INC. — May 11, 2017
43386-573 43386-573 Lupin Pharmaceuticals,Inc. — January 20, 2016
43386-574 43386-574 Lupin Pharmaceuticals,Inc. — November 13, 2015
43386-575 43386-575 Lupin Pharmaceuticals,Inc. — November 13, 2015
75834-324 75834-324 Nivagen Pharmaceuticals, Inc. — April 16, 2024
75834-325 75834-325 Nivagen Pharmaceuticals, Inc. — April 16, 2024
75834-326 75834-326 Nivagen Pharmaceuticals, Inc. — April 16, 2024
43547-486 43547-486 Solco Healthcare US,LLC — July 1, 2020
43547-487 43547-487 Solco Healthcare US,LLC — July 1, 2020
43547-488 43547-488 Solco Healthcare US,LLC — July 1, 2020
0406-1142 0406-1142 SpecGx LLC — November 27, 1998
0406-1144 0406-1144 SpecGx LLC — November 27, 1998
0406-1146 0406-1146 SpecGx LLC — November 27, 1998
57664-228 57664-228 Sun Pharmaceutical Industries, Inc. — August 16, 2013
57664-229 57664-229 Sun Pharmaceutical Industries, Inc. — August 16, 2013
57664-230 57664-230 Sun Pharmaceutical Industries, Inc. — August 16, 2013
72865-122 72865-122 XLCare Pharmaceuticals Inc — February 26, 2020
72865-123 72865-123 XLCare Pharmaceuticals Inc — February 26, 2020
72865-124 72865-124 XLCare Pharmaceuticals Inc — February 26, 2020

Sources for this page

Every dataset that contributed a fact to this page.
Dataset Agency Used for
NDC Directory FDA Identity, ingredients, strengths, forms, routes, labelers, packages
Drugs@FDA FDA Application, sponsor, submissions, review documents, marketing status
Orange Book FDA Therapeutic equivalence codes, reference drug flags, patents, exclusivity
Drug Labeling FDA / NLM Prescribing information reproduced above
FAERS FDA Adverse event report counts
Enforcement FDA Recall records

Generated September 25, 2026 · 13 sections on this page.